2-Acylamino-4, 6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats

2-Acylamino-4, 6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male rats

T Kobayashi, S Sasaki, N Tomita, S Fukui… - Bioorganic & medicinal …, 2010 - Elsevier

GPR54 is a G protein-coupled receptor (GPCR) which was formerly an orphan receptor. Recent
functional study of GPR54 revealed that the receptor plays an essenti.

Peptide synthesis, peptide modification and peptide library synthesis, please contact:

Eva He

eva@pepmic.com

Pepmic Co., Ltd

www.pepmic.com