Molecular design, synthesis, and evaluation of SNIPER (ER) that induces proteasomal degradation of ERα

Molecular design, synthesis, and evaluation of SNIPER (ER) that induces proteasomal degradation of ERα

K Okuhira, Y Demizu, T Hattori, N Ohoka… - … Receptors: Methods and …, 2016 - Springer

... 7. 4-Hydroxytamoxifen (4-OHT): 10–30 μM. 8. Bestatin Methyl Ester (MeBS, Millipore): 10–30
μM. 9. MG-132 (proteasome inhibitor, Z-Leu-Leu-Leu-H (aldehyde)): 10 μM (Peptide Institute).
10. Staurosporine: 1–4 μM. 11. Hydrogen peroxide: 500 μM to 2 mM. 12. ...

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