Internal Peptide Late‐Stage Diversification: Peptide‐Isosteric Triazoles for Primary and Secondary C(sp3)−H Activation
M Bauer, W Wang, MM Lorion, C Dong… - Angewandte Chemie …, 2018 - Wiley Online Library
Abstract Secondary C (sp3)− H arylations were accomplished by palladium catalysis with
triazoles as peptide bond isosteres. The unique power of this approach is highlighted by the
possibility of achieving secondary C (sp3)− H functionalizations on terminal peptides as well …
triazoles as peptide bond isosteres. The unique power of this approach is highlighted by the
possibility of achieving secondary C (sp3)− H functionalizations on terminal peptides as well …
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